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ALK Inhibitor

Product categories of ALK Inhibitor, we are specialized manufacturers from China, Crizotinib Inhibitor, Ap26113 Inhibitor suppliers/factory, wholesale high-quality products of Ceritinib Inhibitor R & D and manufacturing, we have the perfect after-sales service and technical support. Look forward to your cooperation!
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PF-06463922
PF-06463922
Packaging:1g/bag
Biological Activity PF-06463922 demonstrates significant cell activity against ALK and a large set of ALK clinical mutations with IC50 ranging from 0.2 nM-77 nM. [1] PF-06463922 significantly inhibits cell proliferation and induces cell apoptosis in the HCC78 human NSCLC cells harboring SLC34A2-ROS1 fusions and the...
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AP26113
AP26113
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ASP3026
ASP3026
Packaging:1g/bag 1kg/bag
Molecular Weight: 580.74 ASP3026 is a novel and selective inhibitor for ALK with IC50 of 3.5 nM. Phase 1. Biological Activity ASP3026 shows more selective ALK inhibition in a Tyr-kinase panel than PF02341066. ASP3026 inhibits the growth of NCI-H2228, a human NSCLC tumor cell line endogenously expressing EML4-ALK...
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AZD3463
AZD3463
Molecular Weight: 448.95 AZD3463 is a novel orally bioavailable ALK inhibitor with Ki of 0.75 nM, which also inhibits IGF1R with equivalent potency. Biological Activity AZD3463 is potent in ALK-driven preclinical models and in a variety of crizotinib-resistant models. AZD3463 inhibits ALK in cells as demonstrated by...
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AZD3463
AZD3463
Molecular Weight: 448.95 AZD3463 is a novel orally bioavailable ALK inhibitor with Ki of 0.75 nM, which also inhibits IGF1R with equivalent potency. Biological Activity AZD3463 is potent in ALK-driven preclinical models and in a variety of crizotinib-resistant models. AZD3463 inhibits ALK in cells as demonstrated by...
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GSK1838705A
GSK1838705A
Molecular Weight: 532.57 GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein kinases. Biological Activity GSK1838705A potently and ATP-competitively inhibits IGF-1R and IR with appKi values of 0.7...
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Alectinib (CH5424802)
Alectinib (CH5424802)
Molecular Weight: 482.62 Alectinib (CH5424802) is a potent ALK inhibitor with IC50 of 1.9 nM, sensitive to L1196M mutation and higher selectivity for ALK than PF-02341066, NVP-TAE684 and PHA-E429. Biological Activity The dissociation constant (KD) value of CH5424802 for ALK in an ATP-competitive manner is 2.4 nM....
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TAE684 (NVP-TAE684)
TAE684 (NVP-TAE684)
Molecular Weight:614.2 TAE684 is a potent and selective ALK inhibitor with IC50 of 3 nM, 100-fold more sensitive for ALK than InsR. Biological Activity TAE684 does not exhibit significant cross-reactivity against other kinases. TAE684 potently inhibits the proliferation of Ba/F3 NPM-ALK cells with IC50 of 3 nM,...
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Ceritinib (LDK378)
Ceritinib (LDK378)
Brand:Crene
Packaging:1g/bag 1kg/bag
Certificate:GMP
Molecular Weight: 558.14 LDK378 is potent inhibitor against ALK with IC50 of 0.2 nM, shows 40- and 35-fold selectivity against IGF-1R and InsR, respectively. Phase 3. Biological Activity LDK378 shows great anti-proliferative activity in Ba/F3-NPM-ALK and Karpas290 cells with IC50 of 26.0 nM and 22.8 nM, compared with...
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AP26113
AP26113
Molecular Weight: 529.01 AP26113 is a potent ALK inhibitor with IC50 of 0.62 nM, demonstrated ability overcome Crizotinib resistance mediated by a L1196M mutation. Phase 2. Biological Activity AP26113 is highly active against both sensitive and resistant H3122 cells, decreasing cell growth, suppressing ALK...
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GSK1838705A
GSK1838705A
Molecular Weight: 532.57 GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein kinases. Biological Activity GSK1838705A potently and ATP-competitively inhibits IGF-1R and IR with appKi values of 0.7...
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ASP3026
ASP3026
Molecular Weight: 580.74 ASP3026 is a novel and selective inhibitor for ALK with IC50 of 3.5 nM. Phase 1. Biological Activity ASP3026 shows more selective ALK inhibition in a Tyr-kinase panel than PF02341066. ASP3026 inhibits the growth of NCI-H2228, a human NSCLC tumor cell line endogenously expressing EML4-ALK...
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TAE684 (NVP-TAE684)
TAE684 (NVP-TAE684)
.cp_wz table {border-top: 1px solid #ccc;border-left:1px solid #ccc; } .cp_wz table td{border-right: 1px solid #ccc; border-bottom: 1px solid #ccc; padding: 5px 0px 0px 5px;} .cp_wz table th {border-right: 1px solid #ccc;border-bottom: 1px solid #ccc; padding: 5px 0px 0px 5px;} Molecular Weight: 614.2 TAE684 is a...
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Alectinib (CH5424802)
Alectinib (CH5424802)
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GSK1838705A
GSK1838705A
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China ALK Inhibitor Suppliers

ALK Inhibitor

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